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4

Jul

Synthesis, in silico and in vitro evaluation of novel thiazole

  • Project Start Date

    01/07/2018

  • Timeline

    6 month

Synthesis, in silico and in vitro evaluation of novel thiazole and thiadiazole derivatives as multifunctional neurotherapeutic agents.

Computational design, identification of novel lead compounds possessing thiazole/thiadiazole scaffolds and evaluation of their in vitro enzyme inhibition activity on multiple targets, i.e, Monoamine Oxidase-A/B (MAO-A/B) and Acetylcholinesterase (AChE) enzymes.